{"id":6568,"date":"2022-10-21T09:56:56","date_gmt":"2022-10-21T07:56:56","guid":{"rendered":"https:\/\/nanexa.com\/?page_id=6568"},"modified":"2026-09-17T12:59:47","modified_gmt":"2026-09-17T10:59:47","slug":"nex-22","status":"publish","type":"page","link":"https:\/\/nanexa.com\/sv\/nex-22\/","title":{"rendered":"NEX-22"},"content":{"rendered":"\n<div class=\"block-project full-width-container alignfull\">\n\t<div class=\"block-project-list\">\n\t\t<div class=\"block-project-list-left\">\n\t\t\t\t\t\t<div class=\"block-project-list-heading\">\n\t\t\t\t<div class=\"acf-innerblocks-container\">\n\n<h1 id=\"nex-20-for-the-treatment-of-mm\" class=\"wp-block-heading\">NEX-22<\/h1>\n\n\n\n<h2 id=\"nex-20-for-the-treatment-of-mm\" class=\"wp-block-heading\">M\u00e5natliga och kvartalsvisa GLP-1-analoger f\u00f6r behandling av Typ 2-diabetes och fetma <\/h2>\n\n\n\n<h3 id=\"nex-20-for-the-treatment-of-mm\" class=\"wp-block-heading\">Kontrollerad fris\u00e4ttning f\u00f6r f\u00e4rre injektioner<\/h3>\n\n\n\n<p class=\"wp-block-paragraph\">NEX-22 \u00e4r Nanexas program f\u00f6r l\u00e5ngverkande GLP-1 baserat p\u00e5 PharmaShell\u00ae. Efter kliniskt proof of concept med liraglutid en g\u00e5ng i m\u00e5naden \u00e4ndrade Nanexa inriktning till semaglutid f\u00f6r att utveckla m\u00e5natlig och potentiellt kvartalsvis dosering med en j\u00e4mnare farmakokinetisk profil.<\/p>\n\n<\/div>\n\t\t\t<\/div>\n\t\t\t<div class=\"project-list\">\n\t\t\t\t\t\t\t\t\t\t\t\t<ol><li><a href=\"#project-id-1\">Fr\u00e5n liraglutid till semaglutid<\/a><\/li><li><a href=\"#project-id-2\">Vad \u00e4r typ 2-diabetes?<\/a><\/li><li><a href=\"#project-id-3\">B\u00e4ttre efterlevnad och bekv\u00e4mare behandling<\/a><\/li>\t\t\t\t<\/ol>\t\t\t<\/div>\n\t\t<\/div>\n\t\t<div class=\"block-project-list-image\">\n\t\t\t<img decoding=\"async\" src=\"\" style=\"width:100%\">\n\t\t<\/div>\n\t<\/div>\n<\/div>\n\n\n\n<section id=\"project-id-1\" class=\"project-section\"><div class=\"nex-border\"><\/div><div class=\"nex-section-rubrik\"><p>Fr\u00e5n liraglutid till semaglutid<\/p><\/div><div class=\"block-project-heading\"><div class=\"acf-innerblocks-container\">\n\n<p class=\"wp-block-paragraph\">NEX-22-projektet inleddes med en utv\u00e4rdering av PharmaShell\u00ae f\u00f6r liraglutid, en GLP-1 som marknadsf\u00f6rs f\u00f6r daglig administrering.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Den slutf\u00f6rda fas 1-studien gav kliniskt proof of concept: en enda subkutan dos visades uppr\u00e4tth\u00e5lla exponeringen f\u00f6r liraglutid under 36 dagar, med doslinj\u00e4ritet f\u00f6r exponering och Cmax. Den kliniska studien genererade viktiga data fr\u00e5n m\u00e4nniska om fris\u00e4ttningsbeteende, s\u00e4kerhet och tolerabilitet.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Med utg\u00e5ngspunkt i dessa resultat flyttade Nanexa utvecklingsfokus fr\u00e5n liraglutid till semaglutid. Resultaten f\u00f6r liraglutid skapade den kliniska grund och modelleringsgrund som anv\u00e4ndes f\u00f6r att vidareutveckla PharmaShell\u00ae-bel\u00e4ggningarna, f\u00f6rb\u00e4ttra formuleringsstrategin och p\u00e5skynda utvecklingen \u00e4ven av l\u00e5ngverkande semaglutid.<\/p>\n\n\n\n<h2 class=\"wp-block-heading\">Projekt\u00f6verg\u00e5ng<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">Liraglutid etablerade kliniskt proof of concept. Semaglutid \u00e4r nu den GLP-1 som st\u00e5r i fokus och befinner sig f\u00f6r n\u00e4rvarande i preklinisk utveckling. M\u00e5let \u00e4r en differentierad l\u00e5ngverkande GLP-1-analogprodukt med administrering en g\u00e5ng i m\u00e5naden och potentiellt en g\u00e5ng per kvartal.<\/p>\n\n<\/div><\/div><\/section>\n\n<section id=\"project-id-2\" class=\"project-section\"><div class=\"nex-border\"><\/div><div class=\"nex-section-rubrik\"><p>Vad \u00e4r typ 2-diabetes?<\/p><\/div><div class=\"block-project-heading\"><div class=\"acf-innerblocks-container\">\n\n<div class=\"wp-block-columns is-layout-flex wp-container-core-columns-is-layout-8f761849 wp-block-columns-is-layout-flex\">\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\" style=\"flex-basis:60%\">\n<p class=\"wp-block-paragraph\">Typ 2-diabetes \u00e4r en \u00e4mnesoms\u00e4ttningssjukdom d\u00e4r kroppen har sv\u00e5rt att reglera blodsockerniv\u00e5n, vilket leder till h\u00f6gt blodsocker.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Sjukdomen upptr\u00e4der fr\u00e4mst i \u00f6vre medel\u00e5ldern (&gt;45 \u00e5r), men f\u00f6rekomsten \u00f6kar bland yngre personer p\u00e5 grund av en alltmer stillasittande livsstil och oh\u00e4lsosamma matvanor.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Vanliga symtom \u00e4r tr\u00f6tthet, \u00f6kad t\u00f6rst och t\u00e4ta urineringar. Symtomen \u00e4r inledningsvis diffusa och kan ibland vara sv\u00e5ra att uppt\u00e4cka. Typ 2-diabetes kan orsaka flera allvarliga f\u00f6ljdsjukdomar, s\u00e5som njurskador, f\u00f6rs\u00e4mrad syn och hj\u00e4rtsjukdom. Behandling \u00e4r d\u00e4rf\u00f6r avg\u00f6rande, b\u00e5de f\u00f6r patienternas allm\u00e4nna h\u00e4lsa och v\u00e4lbefinnande och f\u00f6r att begr\u00e4nsa de kostnader som sjukdomen medf\u00f6r f\u00f6r h\u00e4lso- och sjukv\u00e5rden och samh\u00e4llet.<\/p>\n<\/div>\n\n\n\n<div class=\"wp-block-column is-vertically-aligned-top is-layout-flow wp-block-column-is-layout-flow\" style=\"flex-basis:33.33%\"><\/div>\n<\/div>\n\n\n\n<h2 class=\"wp-block-heading has-medium-font-size\">F\u00f6rekomst<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">Typ 2-diabetes \u00e4r en av de vanligaste sjukdomarna, och f\u00f6rekomsten \u00f6kar snabbt i takt med en \u00e5ldrande befolkning. Datamonitor Healthcare uppskattar att cirka 600 miljoner m\u00e4nniskor i v\u00e4rlden lever med typ 2-diabetes i dag, en siffra som ber\u00e4knas \u00f6ka till 635 miljoner \u00e5r 2027<sup>(2)<\/sup>.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Av de som lever med typ 2-diabetes blir tyv\u00e4rr inte alla diagnostiserade och antalet som inte f\u00e5r adekvat behandling \u00e4r \u00e4nnu st\u00f6rre. I de sju stora marknaderna i v\u00e4stv\u00e4rlden ber\u00e4knas cirka 50 miljoner personer bli behandlade med l\u00e4kemedel 2027<sup>(1)<\/sup>, med en \u00f6kning p\u00e5 2-3% per \u00e5r.<\/p>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<h2 class=\"wp-block-heading has-medium-font-size\">Behandling<\/h2>\n\n\n<div class=\"\"><img decoding=\"async\" class=\"image-right-float\" src=\"\"><\/div><div><div class=\"acf-innerblocks-container\">\n\n<p class=\"wp-block-paragraph\">M\u00e5let med behandlingen av typ 2-diabetes \u00e4r att s\u00e4nka blodsockerniv\u00e5n. Livsstilsf\u00f6r\u00e4ndringar avseende matvanor och motion \u00e4r ett viktigt f\u00f6rsta steg. En kalorifattig kost och fysisk aktivitet \u00e4r centrala f\u00f6r att s\u00e4nka blodsockerniv\u00e5erna.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Det finns flera l\u00e4kemedel f\u00f6r behandling av typ 2-diabetes. GLP-1-receptoragonister \u00e4r en viktig l\u00e4kemedelsklass och administreras dagligen eller veckovis beroende p\u00e5 den aktiva substansen och formuleringen. Semaglutid marknadsf\u00f6rs f\u00f6r n\u00e4rvarande som en subkutan behandling en g\u00e5ng i veckan, medan Nanexas program syftar till att f\u00f6rl\u00e4nga doseringsintervallet till en g\u00e5ng i m\u00e5naden eller potentiellt en g\u00e5ng per kvartal.<\/p>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<div class=\"wp-block-columns are-vertically-aligned-center break-desktop is-layout-flex wp-container-core-columns-is-layout-8f761849 wp-block-columns-is-layout-flex\">\n<div class=\"wp-block-column is-vertically-aligned-center is-layout-flow wp-block-column-is-layout-flow\">\n<h2 class=\"wp-block-heading has-medium-font-size\">Marknad<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">F\u00f6rs\u00e4ljningen av l\u00e4kemedel mot typ 2-diabetes p\u00e5 de sju st\u00f6rsta marknaderna i v\u00e4stv\u00e4rlden uppskattades till cirka 50 miljarder USD \u00e5r 2022. GLP-1-analoger stod f\u00f6r cirka 15 miljarder USD och f\u00f6rv\u00e4ntades v\u00e4xa med omkring 10 % per \u00e5r under perioden 2022\u20132029<sup>(1)<\/sup>.<\/p>\n<\/div>\n\n\n\n<div class=\"wp-block-column is-vertically-aligned-center is-layout-flow wp-block-column-is-layout-flow\"><\/div>\n<\/div>\n\n<\/div><\/div>\n<\/div><\/div><\/section>\n\n<section id=\"project-id-3\" class=\"project-section\"><div class=\"nex-border\"><\/div><div class=\"nex-section-rubrik\"><p>B\u00e4ttre f\u00f6ljsamhet och smidigare behandling<\/p><\/div><div class=\"block-project-heading\"><div class=\"acf-innerblocks-container\">\n\n<div class=\"wp-block-columns are-vertically-aligned-bottom is-layout-flex wp-container-core-columns-is-layout-8f761849 wp-block-columns-is-layout-flex\">\n<div class=\"wp-block-column is-vertically-aligned-bottom is-layout-flow wp-block-column-is-layout-flow\" style=\"flex-basis:60%\">\n<h2 id=\"controlled-release-increased-compliance\" class=\"wp-block-heading has-medium-font-size\">L\u00e5ngverkande semaglutid<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">NEX-22 fokuserar nu p\u00e5 PharmaShell\u00ae-belagt semaglutid. Formuleringen \u00e4r utformad f\u00f6r att fris\u00e4tta semaglutid kontrollerat under en l\u00e4ngre period, med m\u00e5let att uppr\u00e4tth\u00e5lla en terapeutiskt relevant exponering samtidigt som doseringsfrekvensen minskas och uttalade koncentrationstoppar undviks.<\/p>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<h2 class=\"wp-block-heading has-medium-font-size\">Farmakokinetisk profil<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">Prekliniska data f\u00f6r semaglutid och simuleringar p\u00e5 m\u00e4nniska st\u00f6djer j\u00e4mna exponeringsprofiler vid f\u00f6rl\u00e4ngda doseringsintervall. I internt f\u00f6retagsmaterial fr\u00e5n augusti 2026 redovisar Nanexa simulerade topp\u2013dal-kvoter p\u00e5 1,2 vid dosering en g\u00e5ng i m\u00e5naden och 1,5 vid dosering en g\u00e5ng per kvartal, j\u00e4mf\u00f6rt med 1,8 f\u00f6r marknadsf\u00f6rt semaglutid en g\u00e5ng i veckan. Dessa modellerade profiler st\u00f6djer programmets m\u00e5l om stabil exponering med en l\u00e5g initial topp.<\/p>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<div class=\"wp-block-columns is-layout-flex wp-container-core-columns-is-layout-8f761849 wp-block-columns-is-layout-flex\">\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\" style=\"flex-basis:60%\">\n<figure class=\"wp-block-table\"><table class=\"has-fixed-layout\"><tbody><tr><td><strong>Doseringsprofil<\/strong><\/td><td><strong>Dos<\/strong><\/td><td><strong>Topp\u2013dal-kvot<\/strong><\/td><\/tr><tr><td>Marknadsf\u00f6rt semaglutid, veckovis<\/td><td>2,4 mg<\/td><td>1,8<\/td><\/tr><tr><td>PharmaShell\u00ae-semaglutid, m\u00e5nadsvis<\/td><td>12,3 mg<\/td><td>1,2<\/td><\/tr><tr><td>PharmaShell\u00ae-semaglutid, kvartalsvis<\/td><td>43,7 mg<\/td><td>1,5<\/td><\/tr><\/tbody><\/table><\/figure>\n<\/div>\n<\/div>\n\n\n\n<div class=\"wp-block-columns is-layout-flex wp-container-core-columns-is-layout-8f761849 wp-block-columns-is-layout-flex\">\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\">\n<h3 class=\"wp-block-heading\">M\u00c5NATLIG PK-PROFIL<\/h3>\n\n\n\n<p class=\"wp-block-paragraph\">Simulerad upprepad dosering hos m\u00e4nniska: PharmaShell\u00ae-semaglutid var 28:e dag<\/p>\n\n\n\n<h3 class=\"wp-block-heading\">Stabil exponering \u2022 topp\u2013dal-kvot 1,2<\/h3>\n<\/div>\n\n\n\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\">\n<h3 class=\"wp-block-heading\">KVARTALSVIS PK-PROFIL<\/h3>\n\n\n\n<p class=\"wp-block-paragraph\">Simulerad upprepad dosering hos m\u00e4nniska: PharmaShell\u00ae-semaglutid var 90:e dag<\/p>\n\n\n\n<h3 class=\"wp-block-heading\">F\u00f6rl\u00e4ngd kontroll \u2022 topp\u2013dal-kvot 1,5<\/h3>\n<\/div>\n\n\n\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\"><\/div>\n<\/div>\n<\/div>\n\n\n\n<div class=\"wp-block-column is-vertically-aligned-bottom is-layout-flow wp-block-column-is-layout-flow\">\n<figure class=\"wp-block-image size-full\"><a href=\"https:\/\/nanexa.com\/wp-content\/uploads\/2026\/09\/Nanexa-graf-0917.png\"><img loading=\"lazy\" decoding=\"async\" width=\"946\" height=\"648\" src=\"https:\/\/nanexa.com\/wp-content\/uploads\/2026\/09\/Nanexa-graf-0917.png\" alt=\"Graf \" class=\"wp-image-8190\" srcset=\"https:\/\/nanexa.com\/wp-content\/uploads\/2026\/09\/Nanexa-graf-0917.png 946w, https:\/\/nanexa.com\/wp-content\/uploads\/2026\/09\/Nanexa-graf-0917-300x205.png 300w, https:\/\/nanexa.com\/wp-content\/uploads\/2026\/09\/Nanexa-graf-0917-768x526.png 768w\" sizes=\"auto, (max-width: 946px) 100vw, 946px\" \/><\/a><figcaption class=\"wp-element-caption\">Sammanfattning av PK-profiler baserad p\u00e5 simuleringarna av semaglutid med m\u00e5nadsvis och kvartalsvis dosering. De modellerade resultaten \u00e4r inte kliniska utfall.<\/figcaption><\/figure>\n<\/div>\n<\/div>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<h2 class=\"wp-block-heading has-medium-font-size\">F\u00f6rb\u00e4ttrad f\u00f6ljsamhet genom mindre frekvent dosering<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">L\u00e5ngsiktig behandlingsf\u00f6ljsamhet \u00e4r fortfarande en betydande utmaning vid kronisk GLP-1-behandling. Att f\u00f6rl\u00e4nga doseringsintervallet f\u00f6r semaglutid fr\u00e5n en g\u00e5ng per vecka till en g\u00e5ng var tredje m\u00e5nad har potential att avsev\u00e4rt minska behandlingsb\u00f6rdan och f\u00f6rb\u00e4ttra f\u00f6ljsamheten till behandling.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Programmet syftar till att kombinera s\u00e4llsynta administreringstillf\u00e4llen med kontrollerad fris\u00e4ttning av l\u00e4kemedlet och en l\u00e5g initial toppkoncentration i plasma, egenskaper som kan f\u00f6rb\u00e4ttra tolerabilitet, f\u00f6ljsamhet och l\u00e5ngsiktig kvarstannandegrad i behandling.<\/p>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<h2 class=\"wp-block-heading has-medium-font-size\">Anv\u00e4ndarv\u00e4nlig<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">En l\u00e5ngverkande semaglutidprodukt skulle kunna erbjuda ett differentierat alternativ till dagens veckovisa behandlingar. PharmaShell\u00ae m\u00f6jligg\u00f6r h\u00f6g l\u00e4kemedelsbelastning, l\u00e5g injektionsvolym och kontrollerad fris\u00e4ttning utan att semaglutidmolekylen f\u00f6r\u00e4ndras. M\u00e5lproduktprofilen omfattar dosering en g\u00e5ng i m\u00e5naden eller en g\u00e5ng per kvartal, potential f\u00f6r f\u00f6rvaring i rumstemperatur och kompatibilitet med patientv\u00e4nliga injektionshj\u00e4lpmedel.<\/p>\n\n\n\n<div style=\"height:24px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n\n<div class=\"source\"  style=\"margin:20px -20px\">\n    <div class=\"acf-innerblocks-container\">\n\n<p class=\"wp-block-paragraph\"><strong>(1)<\/strong> Global Data Type 2-diabetes forecast 2021<br><strong>(2)<\/strong> Datamonitor Type 2-diabetes Disease analysis March 2021<\/p>\n\n<\/div>\n<\/div>\n\n<\/div><\/div><\/section>","protected":false},"excerpt":{"rendered":"<p>NEX-22<\/p>\n<p>M\u00e5natliga och kvartalsvisa GLP-1-analoger f\u00f6r behandling av Typ 2-diabetes och fetma <\/p>\n<p>Kontrollerad fris\u00e4ttning f\u00f6r f\u00e4rre injektioner<\/p>\n<p class=\"wp-block-paragraph\">NEX-22 \u00e4r Nanexas program f\u00f6r l\u00e5ngverkande GLP-1 baserat p\u00e5 PharmaShell\u00ae. Efter kliniskt proof of concept med liraglutid en g\u00e5ng i m\u00e5naden \u00e4ndrade Nanexa inriktning till semaglutid f\u00f6r att utveckla m\u00e5natlig och potentiellt kvartalsvis dosering med en j\u00e4mnare farmakokinetisk profil.<\/p>\n<p><a class=\"read-more\" href=\"https:\/\/nanexa.com\/sv\/nex-22\/\">L\u00e4s mer<\/a><\/p>\n","protected":false},"author":1,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":{"_acf_changed":false,"footnotes":""},"class_list":["post-6568","page","type-page","status-publish","hentry"],"acf":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v28.6 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>NEX-22 - Nanexa AB<\/title>\n<meta name=\"description\" content=\"NEX-22 M\u00e5natliga och kvartalsvisa GLP-1-analoger f\u00f6r behandling av Typ 2-diabetes och fetma.\" \/>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/nanexa.com\/sv\/nex-22\/\" \/>\n<meta property=\"og:locale\" content=\"sv_SE\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"NEX-22 - 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